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Optimization of Tubulysin Antibody-Drug-Conjugates: A Case Study in Addressing ADC Metabolism.Tumey, L. Nathan; Leverett, Carolyn A; Vetelino, Beth C.; Li, Fengping; Rago, Brian; Han, Xiaogang; Loganzo, Frank; Musto, Sylvia; Bai, Guoyun; Sukuru, Sai Chetan K; Graziani, Edmund Idris; Puthenveetil, Sujiet; Casavant, Jeffrey; Ratnayake, Anokha Sayani; Marquette, Kimberly; Hudson, Sarah; Doppalapudi, Venkata Ramana; Stock, Joseph R.; Tchistiakova, Lioudmila; Bessire, Andrew J.; Clark, Tracey; Lucas, Judy; Hosselet, Christine; O'Donnell, Christopher J.; Subramanyam, Chakrapani · ACS Medicinal Chemistry Letters · 2016