![Discovery of A Potent and Selective In Vivo Probe (GNE-272) for the Bromodomains of CBP/EP300]()
Discovery of A Potent and Selective In Vivo Probe (GNE-272) for the Bromodomains of CBP/EP300Crawford, Terry D.; Romero, F. Anthony; Lai, Kwong Wah; Tsui, Vickie; Taylor, Alexander M.; de Leon Boenig, Gladys; Noland, Cameron L.; Murray, Jeremy M.; Ly, Justin; Choo, Edna F.; Hunsaker, Thomas L.; Chan, Emily W.; Merchant, Mark; Kharbanda, Samir; Gascoigne, Karen E.; Kaufman, Susan; Beresini, Maureen H.; Liao, Jiangpeng; Liu, Wenfeng; Chen, Kevin X.; Chen, Zhongguo; Conery, Andrew R.; Côté, Alexandre; Jayaram, Hariharan; Jiang, Ying; Kiefer, James R.; Kleinheinz, Tracy; Li, Yingjie; Maher, Jonathan; Pardo, Eneida; Poy, Florence; Spillane, Kerry L; Wang, Fei; Wang, Jian; Wei, Xiaocang; Xu, Zhaowu; Xu, Zhongya; Yen, Ivana; Zawadzke, Laura E.; Zhu, Xiaoyu; Bellon, Steven F.; Cummings, Richard T.; Cochran, Andrea G.; Albrecht, Brian K.; Magnuson, Steven R. · Journal of Medicinal Chemistry · 2016