Replacing alkyl sulfonamide with aromatic sulfonamide in sulfonamide-type RXR agonists favors switch towards antagonist activity
Ken-ichi Morishita; Nobumasa Yakushiji; Fuminori Ohsawa; Kayo Takamatsu; Nobuyasu Matsuura; Makoto Makishima; Masatoshi Kawahata; Kentaro Yamaguchi; Akihiro Tai; Kenji Sasaki; Hiroki Kakuta
- 作者Ken-ichi Morishita; Nobumasa Yakushiji; Fuminori Ohsawa; Kayo Takamatsu; Nobuyasu Matsuura; Makoto Makishima; Masatoshi Kawahata; Kentaro Yamaguchi; Akihiro Tai; Kenji Sasaki; Hiroki Kakuta
- 卷第19卷
- 期第3期
- 印刷ISSN0960-894X
- 文件大小292.75KB
- 发表时间2009
- DOI10.1016/j.bmcl.2008.11.086
- 页码1001-1003