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Pseudo-Cyclization through Intramolecular Hydrogen Bond Enables Discovery of Pyridine Substituted Pyrimidines as New Mer Kinase Inhibitors

Pseudo-Cyclization through Intramolecular Hydrogen Bond Enables Discovery of Pyridine Substituted Pyrimidines as New Mer Kinase Inhibitors

Zhang, Weihe; Zhang, Dehui; Stashko, Michael A.; DeRyckere, Deborah; Hunter, Debra; Kireev, Dmitri; Miley, Michael J.; Cummings, Christopher; Lee, Minjung; Norris-Drouin, Jacqueline; Stewart, Wendy M.; Sather, Susan; Zhou, Yingqiu; Kirkpatrick, Gregory; Machius, Mischa; Janzen, William P.; Earp, H. Shelton; Graham, Douglas K.; Frye, Stephen V.; Wang, Xiaodong
  • 期刊名称Journal of Medicinal Chemistry
  • 作者Zhang, Weihe; Zhang, Dehui; Stashko, Michael A.; DeRyckere, Deborah; Hunter, Debra; Kireev, Dmitri; Miley, Michael J.; Cummings, Christopher; Lee, Minjung; Norris-Drouin, Jacqueline; Stewart, Wendy M.; Sather, Susan; Zhou, Yingqiu; Kirkpatrick, Gregory; Machius, Mischa; Janzen, William P.; Earp, H. Shelton; Graham, Douglas K.; Frye, Stephen V.; Wang, Xiaodong
  • 卷第56卷
  • 期第23期
  • 印刷ISSN0022-2623
  • 电子ISSN1520-4804
  • 文件大小5082.60KB
  • 发表时间2013-12-12
  • DOI10.1021/jm401387j
  • 页码9683-9692
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