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Discovery of Highly Potent, Selective, and Efficacious Small Molecule Inhibitors of ERK1/2

Discovery of Highly Potent, Selective, and Efficacious Small Molecule Inhibitors of ERK1/2

Ren, Li; Grina, Jonas; Moreno, David; Blake, James F.; Gaudino, John J.; Garrey, Rustam; Metcalf, Andrew T.; Burkard, Michael; Martinson, Matthew; Rasor, Kevin; Chen, Huifen; Dean, Brian; Gould, Stephen E.; Pacheco, Patricia; Shahidi-Latham, Sheerin; Yin, Jianping; West, Kristina; Wang, Weiru; Moffat, John G.; Schwarz, Jacob B.
  • 期刊名称Journal of Medicinal Chemistry
  • 作者Ren, Li; Grina, Jonas; Moreno, David; Blake, James F.; Gaudino, John J.; Garrey, Rustam; Metcalf, Andrew T.; Burkard, Michael; Martinson, Matthew; Rasor, Kevin; Chen, Huifen; Dean, Brian; Gould, Stephen E.; Pacheco, Patricia; Shahidi-Latham, Sheerin; Yin, Jianping; West, Kristina; Wang, Weiru; Moffat, John G.; Schwarz, Jacob B.
  • 卷第58卷
  • 期第4期
  • 印刷ISSN0022-2623
  • 电子ISSN1520-4804
  • 文件大小5218.20KB
  • 发表时间2015-02-26
  • DOI10.1021/jm501921k
  • 页码1976-1991
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