Design of Selective Benzoxazepin PI3Kδ Inhibitors Through Control of Dihedral Angles
Safina, Brian Salvatore; Elliott, Richard L; Forrest, Andrew K.; Heald, Robert A.; Murray, Jeremy M.; Nonomiya, Jim; Pang, Jodie; Salphati, Laurent; Seward, Eileen M; Staben, Steven Thomas; Ultsch, Mark; Wei, Binqing; Yang, Wenqian; Sutherlin, Daniel P.
- 期刊名称ACS Medicinal Chemistry Letters
- 作者Safina, Brian Salvatore; Elliott, Richard L; Forrest, Andrew K.; Heald, Robert A.; Murray, Jeremy M.; Nonomiya, Jim; Pang, Jodie; Salphati, Laurent; Seward, Eileen M; Staben, Steven Thomas; Ultsch, Mark; Wei, Binqing; Yang, Wenqian; Sutherlin, Daniel P.
- 印刷ISSN1948-5875
- 电子ISSN1948-5875
- 文件大小702.70KB
- 发表时间2017-08-25
- DOI10.1021/acsmedchemlett.7b00170