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Design of Selective Benzoxazepin PI3Kδ Inhibitors Through Control of Dihedral Angles

Design of Selective Benzoxazepin PI3Kδ Inhibitors Through Control of Dihedral Angles

Safina, Brian Salvatore; Elliott, Richard L; Forrest, Andrew K.; Heald, Robert A.; Murray, Jeremy M.; Nonomiya, Jim; Pang, Jodie; Salphati, Laurent; Seward, Eileen M; Staben, Steven Thomas; Ultsch, Mark; Wei, Binqing; Yang, Wenqian; Sutherlin, Daniel P.
  • 期刊名称ACS Medicinal Chemistry Letters
  • 作者Safina, Brian Salvatore; Elliott, Richard L; Forrest, Andrew K.; Heald, Robert A.; Murray, Jeremy M.; Nonomiya, Jim; Pang, Jodie; Salphati, Laurent; Seward, Eileen M; Staben, Steven Thomas; Ultsch, Mark; Wei, Binqing; Yang, Wenqian; Sutherlin, Daniel P.
  • 印刷ISSN1948-5875
  • 电子ISSN1948-5875
  • 文件大小702.70KB
  • 发表时间2017-08-25
  • DOI10.1021/acsmedchemlett.7b00170
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