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Discovery of Fragment-Derived Small Molecules for In Vivo Inhibition of Ketohexokinase (KHK)

Discovery of Fragment-Derived Small Molecules for In Vivo Inhibition of Ketohexokinase (KHK)

Huard, Kim; Ahn, Kay; Amor, Paul A.; Beebe, David A.; Borzilleri, Kris A; Chrunyk, Boris A.; Coffey, Steven B.; Cong, Yang; Conn, Edward L.; Culp, Jeffrey S.; Dowling, Matthew S.; Gorgoglione, Matthew F.; Gutierrez, Jemy A.; Knafels, John D.; Lachapelle, Erik A.; Pandit, Jayvardhan; Parris, Kevin D.; Perez, Sylvie; Pfefferkorn, Jeffrey A.; Price, David A.; Raymer, Brian; Ross, Trenton T.; Shavnya, Andre; Smith, Aaron C.; Subashi, Timothy A.; Tesz, Gregory; Thuma, Benjamin A.; Tu, Meihua; Weaver, John D.; Weng, Yan; Withka, Jane M.; Xing, Gang; Magee, Thomas V
  • 期刊名称Journal of Medicinal Chemistry
  • 作者Huard, Kim; Ahn, Kay; Amor, Paul A.; Beebe, David A.; Borzilleri, Kris A; Chrunyk, Boris A.; Coffey, Steven B.; Cong, Yang; Conn, Edward L.; Culp, Jeffrey S.; Dowling, Matthew S.; Gorgoglione, Matthew F.; Gutierrez, Jemy A.; Knafels, John D.; Lachapelle, Erik A.; Pandit, Jayvardhan; Parris, Kevin D.; Perez, Sylvie; Pfefferkorn, Jeffrey A.; Price, David A.; Raymer, Brian; Ross, Trenton T.; Shavnya, Andre; Smith, Aaron C.; Subashi, Timothy A.; Tesz, Gregory; Thuma, Benjamin A.; Tu, Meihua; Weaver, John D.; Weng, Yan; Withka, Jane M.; Xing, Gang; Magee, Thomas V
  • 印刷ISSN0022-2623
  • 电子ISSN1520-4804
  • 文件大小1295.08KB
  • 发表时间2017-08-30
  • DOI10.1021/acs.jmedchem.7b00947
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