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Discovery of Potent, Selective and Peripherally Restricted Pan-Trk Kinase Inhibitors for the Treatment of Pain

Discovery of Potent, Selective and Peripherally Restricted Pan-Trk Kinase Inhibitors for the Treatment of Pain

Bagal, Sharan K; Andrews, Mark; Bechle, Bruce M.; Bian, Jianwei; Bilsland, James; Blakemore, David C; Braganza, John; Bungay, Peter J.; Corbett, Matthew S.; Cronin, Ciarán N; Cui, Jingrong Jean; Dias, Rebecca; Flanagan, Neil J; Greasley, Samantha E; Grimley, Rachel; James, Kim; Johnson, Eric; Kitching, Linda; Kraus, Michelle L; McAlpine, Indrawan; Nagata, Asako; Ninkovic, Sacha; Omoto, Kiyoyuki; Scales, Stephanie; Skerratt, Sarah E.; Sun, Jianmin; Tran-Dubé, Michelle; Waldron, Gareth J.; Wang, Fen; Warmus, Joseph S
  • 期刊名称Journal of Medicinal Chemistry
  • 作者Bagal, Sharan K; Andrews, Mark; Bechle, Bruce M.; Bian, Jianwei; Bilsland, James; Blakemore, David C; Braganza, John; Bungay, Peter J.; Corbett, Matthew S.; Cronin, Ciarán N; Cui, Jingrong Jean; Dias, Rebecca; Flanagan, Neil J; Greasley, Samantha E; Grimley, Rachel; James, Kim; Johnson, Eric; Kitching, Linda; Kraus, Michelle L; McAlpine, Indrawan; Nagata, Asako; Ninkovic, Sacha; Omoto, Kiyoyuki; Scales, Stephanie; Skerratt, Sarah E.; Sun, Jianmin; Tran-Dubé, Michelle; Waldron, Gareth J.; Wang, Fen; Warmus, Joseph S
  • 印刷ISSN0022-2623
  • 电子ISSN1520-4804
  • 文件大小2340.43KB
  • 发表时间2018-06-26
  • DOI10.1021/acs.jmedchem.8b00633
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