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N-Thiazolylamide-based free fatty-acid 2 receptor agonists: Discovery, lead optimization and demonstration of off-target effect in a diabetes model

N-Thiazolylamide-based free fatty-acid 2 receptor agonists: Discovery, lead optimization and demonstration of off-target effect in a diabetes model

Hoveyda, Hamid R.; Fraser, Graeme L.; Zoute, Ludivine; Dutheuil, Guillaume; Schils, Didier; Brantis, Cyrille; Lapin, Alexey; Parcq, Julien; Guitard, Sandra; Lenoir, François; Bousmaqui, Mohamed El; Rorive, Sarah; Hospied, Sandrine; Blanc, Sébastien; Bernard, Jérôme; Ooms, Frédéric; McNelis, Joanne C.; Olefsky, Jerrold M.
  • 期刊名称Bioorganic & Medicinal Chemistry
  • 作者Hoveyda, Hamid R.; Fraser, Graeme L.; Zoute, Ludivine; Dutheuil, Guillaume; Schils, Didier; Brantis, Cyrille; Lapin, Alexey; Parcq, Julien; Guitard, Sandra; Lenoir, François; Bousmaqui, Mohamed El; Rorive, Sarah; Hospied, Sandrine; Blanc, Sébastien; Bernard, Jérôme; Ooms, Frédéric; McNelis, Joanne C.; Olefsky, Jerrold M.
  • 印刷ISSN0968-0896
  • 文件大小673.52KB
  • 发表时间2018-9
  • DOI10.1016/j.bmc.2018.09.015
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