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Discovery of a Class of Highly Potent Janus Kinase 1/2 (JAK1/2) Inhibitors Demonstrating Effective Cell-Based Blockade of IL-13 Signaling

Discovery of a Class of Highly Potent Janus Kinase 1/2 (JAK1/2) Inhibitors Demonstrating Effective Cell-Based Blockade of IL-13 Signaling

Zak, Mark; Hanan, Emily J.; Lupardus, Patrick; Brown, David G.; Robinson, Colin; Siu, Michael; Lyssikatos, Joseph P.; Romero, F. Anthony; Zhao, Guiling; Kellar, Terry; Mendonca, Rohan; Ray, Nicholas C.; Goodacre, Simon C.; Crackett, Peter H.; McLean, Neville; Hurley, Christopher A.; Yuen, Po-wai; Cheng, Yun-Xing; Liu, Xiongcai; Liimatta, Marya; Kohli, Pawan Bir; Nonomiya, Jim; Salmon, Gary; Buckley, Gerry; Lloyd, Julia; Gibbons, Paul; Ghilardi, Nico; Kenny, Jane R.; Johnson, Adam
  • 期刊名称Bioorganic & Medicinal Chemistry Letters
  • 作者Zak, Mark; Hanan, Emily J.; Lupardus, Patrick; Brown, David G.; Robinson, Colin; Siu, Michael; Lyssikatos, Joseph P.; Romero, F. Anthony; Zhao, Guiling; Kellar, Terry; Mendonca, Rohan; Ray, Nicholas C.; Goodacre, Simon C.; Crackett, Peter H.; McLean, Neville; Hurley, Christopher A.; Yuen, Po-wai; Cheng, Yun-Xing; Liu, Xiongcai; Liimatta, Marya; Kohli, Pawan Bir; Nonomiya, Jim; Salmon, Gary; Buckley, Gerry; Lloyd, Julia; Gibbons, Paul; Ghilardi, Nico; Kenny, Jane R.; Johnson, Adam
  • 印刷ISSN0960-894X
  • 文件大小1954.28KB
  • 发表时间2019-4
  • DOI10.1016/j.bmcl.2019.04.008
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