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TAS4464, a highly potent and selective inhibitor of NEDD8 activating enzyme, suppresses neddylation and shows antitumor activity in diverse cancer models

TAS4464, a highly potent and selective inhibitor of NEDD8 activating enzyme, suppresses neddylation and shows antitumor activity in diverse cancer models

Yoshimura, Chihoko; Muraoka, Hiromi; Ochiiwa, Hiroaki; Tsuji, Shingo; Hashimoto, Akihiro; Kazuno, Hiromi; Nakagawa, Fumio; Komiya, Yu; Suzuki, Satoshi; Takenaka, Toru; Kumazaki, Masafumi; Fujita, Naoya; Mizutani, Takashi; Ohkubo, Shuichi
  • 期刊名称Molecular Cancer Therapeutics
  • 作者Yoshimura, Chihoko; Muraoka, Hiromi; Ochiiwa, Hiroaki; Tsuji, Shingo; Hashimoto, Akihiro; Kazuno, Hiromi; Nakagawa, Fumio; Komiya, Yu; Suzuki, Satoshi; Takenaka, Toru; Kumazaki, Masafumi; Fujita, Naoya; Mizutani, Takashi; Ohkubo, Shuichi
  • 印刷ISSN1535-7163
  • 电子ISSN1538-8514
  • 文件大小1493.34KB
  • 发表时间2019-05-15
  • DOI10.1158/1535-7163.MCT-18-0644
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