Discovery of BMS-986251: A Clinically Viable, Potent, and Selective RORγt Inverse Agonist

• 期刊名称ACS Medicinal Chemistry Letters
• 作者Cherney, Robert J.; Cornelius, Lyndon A. M.; Srivastava, Anurag; Weigelt, Carolyn A.; Marcoux, David; Duan, James J.-W.; Shi, Qing; Batt, Douglas G.; Liu, Qingjie; Yip, Shiuhang; Wu, Dauh-Rurng; Ruzanov, Max; Sack, John; Khan, Javed; Wang, Jinhong; Yarde, Melissa; Cvijic, Mary Ellen; Mathur, Arvind; Li, Sha; Shuster, David; Khandelwal, Purnima; Borowski, Virna; Xie, Jenny; Obermeier, Mary; Fura, Aberra; Stefanski, Kevin; Cornelius, Georgia; Tino, Joseph A.; Macor, John E.; Salter-Cid, Luisa; Denton, Rex; Zhao, Qihong; Carter, Percy H.; Dhar, T. G. Murali
• 印刷ISSN1948-5875
• 电子ISSN1948-5875
• 文件大小526.45KB
• 发表时间2020-04-10
• DOI10.1021/acsmedchemlett.0c00063