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N-Thiazolylamide-based free fatty-acid 2 receptor agonists: Discovery, lead optimization and demonstration of off-target effect in a diabetes modelHoveyda, Hamid R.; Fraser, Graeme L.; Zoute, Ludivine; Dutheuil, Guillaume; Schils, Didier; Brantis, Cyrille; Lapin, Alexey; Parcq, Julien; Guitard, Sandra; Lenoir, François; Bousmaqui, Mohamed El; Rorive, Sarah; Hospied, Sandrine; Blanc, Sébastien; Bernard, Jérôme; Ooms, Frédéric; McNelis, Joanne C.; Olefsky, Jerrold M. · Bioorganic & Medicinal Chemistry · 2018